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AHR antagonist 2

CAS No. 2338747-54-7

AHR antagonist 2( —— )

Catalog No. M32773 CAS No. 2338747-54-7

AHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.

Purity : >98% (HPLC)

COA

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HNMR

HPLC

MSDS

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Biological Information

Product Name

AHR antagonist 2
Note

Research use only, not for human use.
Brief Description

AHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.
Description

AHR antagonist 2 is a potent aryl hydrocarbon receptor (AHR) antagonist, extracted from patent WO2019101641A1, compound example 1, with IC50s of 0.885 and 2.03 nM for human and mouse AhR.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

Aryl Hydrocarbon Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

2338747-54-7
Formula Weight

418.37
Molecular Formula

C20H17F3N4O3
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 250 mg/mL (597.56 mM; Ultrasonic )
SMILES

C[C@@H](CO)NC(=O)c1cc(nc(n1)-c1cccnc1)-c1ccc(OC(F)(F)F)cc1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Julien LEFRANC, et al. 2-hetarylpyrimidine-4-carboxamides as aryl hydrocarbon receptor anatgonists. WO2019101641A1.

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